Journal of Medicinal Chemistry p. 1124 - 1135 (2013)
Update date:2022-09-26
Topics:
Kawasuji, Takashi
Johns, Brian A.
Yoshida, Hiroshi
Weatherhead, Jason G.
Akiyama, Toshiyuki
Taishi, Teruhiko
Taoda, Yoshiyuki
Mikamiyama-Iwata, Minako
Murai, Hitoshi
Kiyama, Ryuichi
Fuji, Masahiro
Tanimoto, Norihiko
Yoshinaga, Tomokazu
Seki, Takahiro
Kobayashi, Masanori
Sato, Akihiko
Garvey, Edward P.
Fujiwara, Tamio
This work is a continuation of our initial discovery of a potent monocyclic carbamoyl pyridone human immunodeficiency virus type-1 (HIV-1) integrase inhibitor that displayed favorable antiviral and pharmacokinetic properties. We report herein a series of
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