Journal of Medicinal Chemistry p. 4442 - 4455 (2013)
Update date:2022-08-15
Topics:
Monn, James A.
Valli, Matthew J.
Massey, Steven M.
Hao, Junliang
Reinhard, Matthew R.
Bures, Mark G.
Heinz, Beverly A.
Wang, Xushan
Carter, Joan H.
Getman, Brian G.
Stephenson, Gregory A.
Herin, Marc
Catlow, John T.
Swanson, Steven
Johnson, Bryan G.
McKinzie, David L.
Henry, Steven S.
As part of our ongoing interest in identifying novel agonists acting at metabotropic glutamate (mGlu) 2/3 receptors, we have explored the effect of structural modifications of 1S,2S,5R,6S-2-aminobicyclo[3.1.0]hexane-2,6- dicarboxylate (LY354740), a potent
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