Azulene derivatives as TXA2/PGH2 receptor antagonists - II. Synthesis and biological activity of 6-mono- and 6-dihydroxylated-isopropylazulenes

DOI: 10.1016/0968-0896(96)00038-7

Source and publish data:

Bioorganic and Medicinal Chemistry p. 575 - 591 (1996)

Update date:2022-07-30

Topics:

Authors:

Yokota, Masayuki

Uchibori, Satoko

Hayashi, Hiromi

Koyama, Rei

Kosakai, Kazuhiro

Wakabayashi, Shuichi

Tomiyama, Tsuyoshi

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0968-0896(96)00038-7

In order to examine the correlation between activity and hydrophilicity of the side chain of sodium 3-[4-(4-chlorobenzenesulfonylamino)butyl]-6- isopropylazulene-1-sulfonate (KT2-962), a non-prostanoid TXA₂/PGH₂ receptor antagonist,

Full text of DOI:10.1016/0968-0896(96)00038-7

Products guided by the article

Product name:3-(4-Benzenesulfonylamino-butyl)-6-isopropyl-azulene-1-sulfonic acid butyl ester

Cas No:150094-27-2

R&D Labs maybe for 150094-27-2

Sinoway Industrial Co., Ltd.

website:http://www.china-sinoway.com

Contact:+86-592-5853819

Address:16/F,Huicheng Comm,Complex,No839 XiaHe Rd, Xiamen,China
Shandong united-rising pharmaceutical cooperation.,ltd.

Contact:008653187965009

Address:171No., Jing5 Road, Shizhong District, Jinan, China
Shenzhen ZheYi Chemicals Co.,LTD(Shanghai Branch)

Contact:+86-21-54159691

Address:Room1002,Building No.2, Lane 98 Bixiu Road,Minhang District, Shanghai,China 201100
Weifang Ocean Trading Co., Ltd.

Contact:+86-536-2081155

Address:Room2606, Yuqing Building, 518#, Yuquan Road, High-tech Development Zone, Weifang City, Shandong Province, China
QUZHOU ZIO I/E CO.;LTD

Contact:13357117572

Address:No.149 Shiji dadao Road.

Relevant to this article

A - And B -fluorinated aminophosphonates-Synthesis and properties

Doi:10.1080/10426507.2015.1091832
(2016)
A series of penicillin derived C2-symmetric inhibitors of HIV-1 proteinase: synthesis, mode of interaction, and structure-activity relationships.

Doi:10.1021/jm00073a011
(1993)
Graphene oxide: An efficient and reusable carbocatalyst for aza-Michael addition of amines to activated alkenes

Doi:10.1039/c1cc15230k
(2011)
Direct detection of S-palmitoylation by mass spectrometry

Doi:10.1021/ac402850s
(2013)
Borole derivatives X. Syntheses of (η⁵-borole)metal complexes via borole ammonia adducts. Complexes of the chromium group metals and the crystal and molecular structures of tetracarbonyl <η⁵-(1-phenylborole)>chromium and its molybden

Doi:10.1016/0022-328X(87)87155-3
(1987)
Oxoammonium Salts. 5. A New Synthesis of Hindered Piperidines Leading to Unsymmetrical TEMPO-Type Nitroxides. Synthesis and Enantioselective Oxidations with Chiral Nitroxides and Chiral Oxoammonium Salts

Doi:10.1021/jo00070a018
(1993)

Article Doi