The dolastatins. 22. Synthesis of Boc-dolaproinyl-dolaphenine and four related chiral isomers

DOI: 10.1021/jo00090a009

Source and publish data:

Journal of Organic Chemistry p. 2935 - 2938 (1994)

Update date:2022-08-03

Topics:

Authors:

Pettit Pettit

Barkoczy

Srirangam

Singh Singh

Herald Herald

Williams

Kantoci Kantoci

Hogan Hogan

Groy Groy

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Article abstract of DOI:10.1021/jo00090a009

Synthesis of the dolastatin 10 (1) dipeptide segment N-(tert-butoxycarbonyl)-dolaproinyl-dolaphenine (2, Boc-Dap-Doe) and four chiral isomers (3-5, 13) has been summarized. Formation of the amide bond was readily accomplished employing diethyl cyanophosph

Full text of DOI:10.1021/jo00090a009

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