Regioselective syntheses of 3-aminomethyl-5-substituted isoxazoles: A facile and chemoselective reduction of azide to amino by sodium borohydride using 1,3-propanedithiol as a catalyst

DOI: 10.1016/S0040-4039(00)60386-6

Source and publish data:

Tetrahedron Letters p. 7509 - 7512 (1993)

Update date:2022-08-02

Topics:

Authors:

Pei Pei

Wickhan Wickhan

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(00)60386-6

A series of isoxazole azides were reduced selectively to isoxazole amines in quantitative yield by sodium borohydride using 1,3-propanedithiol as a catalyst.

Full text of DOI:10.1016/S0040-4039(00)60386-6

Products guided by the article

Product name:1-(5-isopropylisoxazol-3-yl)methanamine

Cas No:154016-49-6

R&D Labs maybe for 154016-49-6

Changsha Huajing Powdery Material Technological Co., Ltd.

Contact:86-731-88879686

Address:Building 2, West Garden, Main Campus of Central South University, Changsha, Hunan Province, China
Jinhua Haoyuan Chemical CO., LTD(expird)

Contact:86-579-82465583

Address:Jinhua,Zhejiang
QINGDAO HONG JIN CHEMICAL CO.,LTD.

website:http://www.hongjinchem.com

Contact:+86-532-83657313

Address:2ND Building, 8 Shangqing Road, Qingdao, Shandong Province, China.
SPRING CHEMICAL INDUSTRY CO.,LTD

Contact:86-187-66672125

Address:linchi industry park.zouping
Henan Surface Industry Co Ltd

Contact:86-371-86169316

Address:No.1,Shakou Road,Zhengzhou,China

Relevant to this article

Targeted theranostic platinum(IV) prodrug with a built-in aggregation-induced emission light-up apoptosis sensor for noninvasive early evaluation of its therapeutic responses in situ

Doi:10.1021/ja411811w
(2014)
A-ring modified steroidal azoles retaining similar potent and slowly reversible CYP17A1 inhibition as abiraterone

Doi:10.1016/j.jsbmb.2014.01.013
(2014)
Novel Steroidal Inhibitors of Human Cytochrome P450_17α (17α-Hydroxylase-C_17,20-lyase): Potential Agents for the Treatment of Prostatic Cancer

Doi:10.1021/jm00013a022
(1995)
A new entry to β-hydroxyphosphonates: The SmI₂-mediated reaction of diethyl iodomethylphosphonate with carbonyl compounds

Doi:10.1016/S0040-4039(02)01539-3
(2002)
Synthesis and structure characterization of homoleptic lanthanide complexes stabilized by Schiff-base ligands and their application in the polymerization of ε-caprolactone

Doi:10.1016/j.jorganchem.2017.12.002
(2018)
N-Arylation of Amino Acid Esters to Expand Side Chain Diversity in Ketoxime Peptide Ligations

Doi:10.1021/acs.joc.9b02810
(2020)

Article Doi