Regioselective syntheses of 3-aminomethyl-5-substituted isoxazoles: A facile and chemoselective reduction of azide to amino by sodium borohydride using 1,3-propanedithiol as a catalyst

DOI: 10.1016/S0040-4039(00)60386-6

Source and publish data:

Tetrahedron Letters p. 7509 - 7512 (1993)

Update date:2022-08-02

Topics:

Authors:

Pei Pei

Wickhan Wickhan

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(00)60386-6

A series of isoxazole azides were reduced selectively to isoxazole amines in quantitative yield by sodium borohydride using 1,3-propanedithiol as a catalyst.

Full text of DOI:10.1016/S0040-4039(00)60386-6

Products guided by the article

Product name:1-(5-isopropylisoxazol-3-yl)methanamine

Cas No:154016-49-6

R&D Labs maybe for 154016-49-6

PINGYUAN SIHUAN PHARMACEUTICAL CO., LTD

Contact:+86-531-55696072

Address:#2766,yinxiu Road, Economic Development Zone, Pingyuan Country, Shandong Province, China.
NOVASYNCS CO., LTD

Contact:0512-63006287

Address:no.88.YISHENG Road,etdz-WUJIANG,SUZHOU,CHINA
ZHUHAI HAIRUIDE BIOSCIENCE AND TECHNOLOGY CO.,LTD

website:http://www.zhhairuide.com

Contact:+8613326687259/+86-756-7789199

Address:No.10 Yonghui Road
Zhejiang Hoshine Silicon Industry Co., Ltd.

Contact:86-573-89179966

Address:Zhapu Town, Pinghu City, Zhejiang, China
Jiangxi Province Bethel Pharmaceutical Co., Ltd.

Contact:+86-795-259 3456 ，+86-15957688008 13566650571

Address:Huangjindui Chemical Park， Shanggao County ，Yichun city，Jiangxi Province

Relevant to this article

Targeted theranostic platinum(IV) prodrug with a built-in aggregation-induced emission light-up apoptosis sensor for noninvasive early evaluation of its therapeutic responses in situ

Doi:10.1021/ja411811w
(2014)
A-ring modified steroidal azoles retaining similar potent and slowly reversible CYP17A1 inhibition as abiraterone

Doi:10.1016/j.jsbmb.2014.01.013
(2014)
Novel Steroidal Inhibitors of Human Cytochrome P450_17α (17α-Hydroxylase-C_17,20-lyase): Potential Agents for the Treatment of Prostatic Cancer

Doi:10.1021/jm00013a022
(1995)
A new entry to β-hydroxyphosphonates: The SmI₂-mediated reaction of diethyl iodomethylphosphonate with carbonyl compounds

Doi:10.1016/S0040-4039(02)01539-3
(2002)
Synthesis and structure characterization of homoleptic lanthanide complexes stabilized by Schiff-base ligands and their application in the polymerization of ε-caprolactone

Doi:10.1016/j.jorganchem.2017.12.002
(2018)
N-Arylation of Amino Acid Esters to Expand Side Chain Diversity in Ketoxime Peptide Ligations

Doi:10.1021/acs.joc.9b02810
(2020)

Article Doi