Regioselective syntheses of 3-aminomethyl-5-substituted isoxazoles: A facile and chemoselective reduction of azide to amino by sodium borohydride using 1,3-propanedithiol as a catalyst

DOI: 10.1016/S0040-4039(00)60386-6

Source and publish data:

Tetrahedron Letters p. 7509 - 7512 (1993)

Update date:2022-08-02

Topics:

Authors:

Pei Pei

Wickhan Wickhan

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Article abstract of DOI:10.1016/S0040-4039(00)60386-6

A series of isoxazole azides were reduced selectively to isoxazole amines in quantitative yield by sodium borohydride using 1,3-propanedithiol as a catalyst.

Full text of DOI:10.1016/S0040-4039(00)60386-6

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