Chemical and Pharmaceutical Bulletin p. 1378 - 1386 (1993)
Update date:2022-08-05
Sakurai
Higashida
Sugano
Nishi
Saito
Ohata
Handa
Komai
Yagi
Nishigaki
Yabe
Human immunodeficiency virus type 1 (HIV-1) protease inhibitors containing four types of hydroxyethylene dipeptide isosteres were designed and synthesized. These inhibitors consist of eight stereoisomers of phenylalanylproline (Phe-Ψ[H.E.]-Pro), four ster
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