In vitro membrane permeation studies and in vivo antinociception of glycosylated Dmt1-DALDA analogues

DOI: 10.1021/ml4004765

Source and publish data:

ACS Medicinal Chemistry Letters p. 352 - 357 (2014)

Update date:2022-08-04

Topics:

Authors:

Ballet, Steven

Betti, Cecilia

Novoa, Alexandre

Toemboely, Csaba

Uhd Nielsen, Carsten

Helms, Hans Christian

Lesniak, Anna

Kleczkowska, Patrycja

Chung, Nga N.

Lipkowski, Andrzej W.

Brodin, Birger

Tourwe, Dirk

Schiller, Peter W.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/ml4004765

In this study the μ opioid receptor (MOR) ligands DALDA (Tyr-d-Arg-Phe-Lys-NH₂) and Dmt¹-DALDA (Dmt-d-Arg-Phe-Lys-NH₂, Dmt = 2′,6′-dimethyltyrosine) were glycosylated at the N- or C-terminus. Subsequently, the modified pep

Full text of DOI:10.1021/ml4004765

Products guided by the article

Product name:C₃₁H₄₂N₈O₅

Cas No:1558028-91-3

R&D Labs maybe for 1558028-91-3

Shandong General Materials Co.,Ltd（Shandong Aoertong Chemical Co., Ltd）

Contact:86-531-88072280

Address:No. 1825 Hualong Road, Licheng District, Jinan, Shandong, China
Shijiazhuang Sdyano Fine Chemical Co., Ltd

Contact:+86-311-89830448

Address:NO.48 Ta Nan Road,Yuhua District,Shijiazhuang,Hebei,China
SHANDONG ZHANHUA YONGHAO PHARMACEUTICAL TECH.CO.,LTD

Contact:+86-576-88685096

Address:GENGJU VILLAGE NORTH ONE KILOMETER,ZHANHUA DISTRICT,BINZHOU CITY,SHANDONG PROVINCE,CHINA.
Guangzhou Swan Chemical Co., Ltd.

Contact:+86-20-31075659

Address:NO.301, Hong ba fang investment BLDG 1,Guan chong village,Shiqi town,Panyu district,Guangzhou
Shanxi Sanwei Group Co.,Ltd

Contact:0086-357-6662688

Address:Zhaocheng town, Hongtong County, Linfen City, Shanxi Province

Relevant to this article

Synthesis and oxidative activation of an oxabicyclo[7.2.1] enediyne

Doi:10.1016/S0040-4020(01)80628-1
(1994)
Efficient and Reusable Pb(II) Metal–Organic Framework for Knoevenagel Condensation

Doi:10.1007/s10562-018-2471-8
(2018)
Design and synthesis of calcium and magnesium ionophores based on double-armed diazacrown ether compounds and their application to an ion-sensing component for an ion-selective electrode

Doi:10.1021/ac00098a016
(1995)
Conversion of 1-(ω-Alkynyl)-1,2-propadienyl Sulfides to Bicyclic Dienones by the Use of Iron Carbonyl Complex

Doi:10.1246/cl.1994.315
(1994)
The effect of molecular planarity on crystal non-centrosymmetry in benzylidene-aniline derivatives

Doi:10.1107/S0108270102006479
(2002)
Nitrile-containing phenolic glucosides from the leaves of Glochidion acuminatum

Doi:10.1248/cpb.c14-00638
(2015)

Article Doi