A Practical Alternative to Sulfonyl Activation of Aziridines: Ring-Opening of N-Diphenylphosphinoyl Aziridines by Carbon Nucleophiles

DOI: 10.1016/S0040-4039(00)77020-1

Source and publish data:

Tetrahedron Letters p. 2739 - 2742 (1994)

Update date:2022-08-03

Topics:

Authors:

Osborn, Helen M. I.

Sweeney, J. B.

Howson, William

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Article abstract of DOI:10.1016/S0040-4039(00)77020-1

The ring-opening reaction of N-diphenylphosphinoylaziridines by Copper (I)-modified Grignard reagents proceeds in good to excellent yield and with complete regiospecificity.

Full text of DOI:10.1016/S0040-4039(00)77020-1

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