Room-temperature Cu(ii)-catalyzed aromatic C-H azidation for the synthesis of ortho-azido anilines with excellent regioselectivity

DOI: 10.1039/c4cc01481b

Source and publish data:

Chemical Communications p. 5733 - 5736 (2014)

Update date:2022-08-04

Topics:

Authors:

Fan, Yunpeng

Wan, Wen

Ma, Guobin

Gao, Wei

Jiang, Haizhen

Zhu, Shizheng

Hao, Jian

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Article abstract of DOI:10.1039/c4cc01481b

Cu(ii)-catalyzed aromatic C-H azidation with azido-benziodoxolone under mild conditions has been described. The primary amine exhibits an excellent ortho-directing effect, providing ortho-azidated anilines as the sole products. the Partner Organisations 2014.

Full text of DOI:10.1039/c4cc01481b

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