
Chemical and Pharmaceutical Bulletin p. 960 - 965 (1995)
Update date:2022-08-03
Topics:
Kiyama
Hayashi
Hara
Fujimoto
Kawabata
Kawakami
Nakajima
Fujishita
A novel series of 6-alkyl-7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxylic acid derivatives was prepared as angiotensin II (AII) receptor antagonists. When evaluated in an in vitro binding assay using COS cells transfected with a cDNA encoding a hu
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