
Journal of Medicinal Chemistry p. 1462 - 1472 (1995)
Update date:2022-09-26
Topics:
Cristalli, Gloria
Camaioni, Emidio
Vittori, Sauro
Volpini, Rosaria
Borea, Pier Andrea
et al.
A series of new 2-aralkynyl and 2-heteroaralkynyl derivatives of NECA were synthesized and studied in binding and functional assays to assess their potency for the A2a compared to A1 adenosine receptors.Compounds bearing an aromatic
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