Journal of Medicinal Chemistry p. 1720 - 1735 (1995)
Update date:2022-08-05
Topics: Structure-activity relationships Chemical Synthesis High-Throughput Screening Structure-activity relationship study Radioligand Binding Assay
Jacobson, Kenneth A.
Siddiqi, Suhaib M.
Olah, Mark E.
Ji, Xiao-duo
Melman, Neli
et al.
9-Alkyladenine derivatives and ribose-modified N6-benzyladenosine derivatives were synthesized in an effort to identify selective ligands for the rat A3 adenosine receptor and leads for the development of antagonists.The derivatives
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