Chemical and Pharmaceutical Bulletin p. 424 - 426 (1997)
Update date:2022-08-03
Topics:
Endo, Yasuyuki
Ohno, Michihiro
Takehana, Shunji
Driedger, Paul E.
Stabel, Silvia
Shudo, Koichi
We synthesized benzolactams with hydrophobic substituents at various positions as analogs of (-)-benzolactam-V8-310 ((-)-BL-V8-310, 1) which reproduces the active conformation and biological activity of teleocidins. Structure-activity data indicate that the existence of a hydrophobic region between C-2 and C-9, and the steric factor at C-8 play critical roles in the appearance of biological activities.
View MoreYingkou Sanzheng Organic Chemical Co. Ltd.
Contact:+86-417-3638818
Address:25 Gengxinli Village, Daqing Road, Yingkou, Liaoning, China
website:https://sdjingyuan.lookchem.com/
Contact:86-531-82687998
Address:Factory Building 11, Jinan Comprehensive free trade zone, Shandong, China
Beijing Century Richap Chemistry Co.,Ltd
Contact:+86- 010-64455497
Address:Guannan County, Lianyungang City, Jiangsu Province, China
Jiangxi Lanqi Fine Chemical S&T Co., Ltd.
Contact:+86-21-64891143
Address:XinJiShan Industrial Area, Zhangshu City, JiangXi Province, China
Shanghai Korey Pharm Co.,Ltd.(expird)
Contact:021-61840961 021-61840962
Address:No.157,Zhuguang Rd, Qingpu, Shanghai, China
Doi:10.1016/0040-4020(95)00511-6
(1995)Doi:10.1039/c5cy01722j
(2016)Doi:10.1016/0020-1693(95)04638-P
(1995)Doi:10.1039/DT9950003019
(1995)Doi:10.1139/v97-146
(1997)Doi:10.3390/molecules15020824
(2010)
