A Direct Route to the Pyrrolobenzodiazepine Ring System Using Aryl Triflates

DOI: 10.1016/0040-4039(95)01592-6

Source and publish data:

Tetrahedron Letters p. 7595 - 7598 (1995)

Update date:2022-08-04

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Authors:

Kraus, George A.

Liu, Peng

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Article abstract of DOI:10.1016/0040-4039(95)01592-6

The pyrrolo<2,1-c><1,4>benzodiazepine and dibenzo<1,4>diazepine skeletons were rapidly generated from salicylic acids.The key step in these syntheses was the substitution of an aryl triflate.

Full text of DOI:10.1016/0040-4039(95)01592-6

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