Diastereoselective synthesis of merucathin: The singlet oxygen ene reaction (Schenck reaction) as a key step towards an E-configured β-amino allylic alcohol

DOI: 10.1055/s-1995-4071

Source and publish data:

Synthesis p. 1066 - 1068 (1995)

Update date:2022-08-02

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Authors:

Adam Adam

Brunker Brunker

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Article abstract of DOI:10.1055/s-1995-4071

An enantio- and diastereoselective synthesis of the naturally occurring merucathin is reported. The singlet oxygen ene reaction of the bis-Boc-protected allylic amine 3, which was prepared from L-alanine, was employed as key step for this regio- and diast

Full text of DOI:10.1055/s-1995-4071

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