Structure-activity relationships of non-peptide vasopressin V(1a) antagonists: 1-(1-multi-substituted benzoyl 4-piperidyl)-3,4-dihydro-2(1H)- quinolinones

DOI: 10.1248/cpb.44.725

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 725 - 733 (1996)

Update date:2022-08-05

Topics:

Authors:

Kondo Kondo

Ogawa Ogawa

Nakaya Nakaya

Tominaga

Yabuuchi

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Article abstract of DOI:10.1248/cpb.44.725

During our systematic studies on the arginine vasopressin receptor V(1a)- antagonistic activity of 1-(1-benzoyl substituted 4-piperidyl)-3,4-dihydro- 2(1H)-quinolinones, we found a general substituent effect on the benzene ring. Hydrogen-bonding ability a

Full text of DOI:10.1248/cpb.44.725

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