Structure-activity relationships of non-peptide vasopressin V(1a) antagonists: 1-(1-multi-substituted benzoyl 4-piperidyl)-3,4-dihydro-2(1H)- quinolinones

DOI: 10.1248/cpb.44.725

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 725 - 733 (1996)

Update date:2022-08-05

Topics:

Authors:

Kondo Kondo

Ogawa Ogawa

Nakaya Nakaya

Tominaga

Yabuuchi

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1248/cpb.44.725

During our systematic studies on the arginine vasopressin receptor V(1a)- antagonistic activity of 1-(1-benzoyl substituted 4-piperidyl)-3,4-dihydro- 2(1H)-quinolinones, we found a general substituent effect on the benzene ring. Hydrogen-bonding ability a

Full text of DOI:10.1248/cpb.44.725

NII-Electronic Library Service

Products guided by the article

Product name:4-(Benzyloxycarbonyl-methyl-amino)-2-methoxy-benzoic acid

Cas No:176547-20-9

R&D Labs maybe for 176547-20-9

Okeanos Tech.Co.,LTD

Contact:+86-10-62651721

Address:29 Yongxing Road, Daxing District,Beijing China
Jingzhou TianHe Sci&Tech Chemical Co., Ltd.

Contact:86-716-8331612

Address:Jiangjin Road, #18, High-grade technology industries development district, Jingzhou city, Hubei province
Hangzhou Gangjin Chemical Co.,Ltd.(expird)

Contact:+86-571-85109780

Address:707 Zhejiang Minhang Bldg., No.290 Zhongshan North Road, Hangzhou 310003, China
Xinchang Yueding Chemical Co., Ltd.

Contact:86-571-56926323

Address:NO.90 BEIMENCHENGWAI CHENGGUAN TOWN XINCHANG
HAORUI ENTERPRISES LLC

Contact:(1) 206-3550089

Address:5115 NE 8TH PL, Renton, WA 98059 USA

Relevant to this article

Synthesis and evaluation of inhibitors of transthyretin amyloid formation based on the non-steroidal anti-inflammatory drug, flufenamic acid

Doi:10.1016/S0968-0896(99)00066-8
(1999)
D-Xylose derived oxazolidin-2-ones as chiral auxiliaries in stereoselective acylations and halogenations

Doi:10.1016/S0957-4166(96)00478-8
(1997)
Doi:10.1515/znb-1996-0217
(1996)
Doi:10.1021/jo01017a021
(1965)
Synthesis and characterization of organomolybdenum and organotungsten halides containing the η⁵-pentaphenylcyclopentadienyl ligand η⁵-C₅Ph₅Mo(CO)₃X·nCH ₂Cl₂ and η⁵-C₅Ph₅W(CO)₃X (X=C1, Br, I).

Doi:10.1016/0020-1693(95)04788-3
(1996)
Total asymmetric synthesis of the potent immunosuppressive marine natural product microcolin A

Doi:10.1021/jo952123l
(1996)

Article Doi