Bioorganic and Medicinal Chemistry Letters p. 2669 - 2674 (1998)
Update date:2022-08-04
Topics:
Muller, George W.
Shire, Mary G.
Wong, Lu Min
Corral, Laura G.
Patterson, Rebecca T.
Chen, Yuxi
Stirling, David I.
N-Phthaloyl 3-amino-3-arylpropionic acid analogs of thalidomide that are potent inhibitors of tumor necrosis factor-α are reported. These compounds were found to be potent inhibitors of phosphodiesterase 4.
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