A new method for the solution and solid phase synthesis of chiral β-sulfonopeptides under mild conditions

DOI: 10.1016/0040-4039(96)01963-6

Source and publish data:

Tetrahedron Letters p. 8589 - 8592 (1996)

Update date:2022-08-05

Topics:

Authors:

Gude, Markus

Piarulli, Umberto

Potenza, Donatella

Salom, Barbara

Gennari, Cesare

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Article abstract of DOI:10.1016/0040-4039(96)01963-6

Chiral β-sulfonopeptides were synthesized both in solution and in the solid phase using the sulfonyl chlorides derived from enantiomerically pure 2-substituted taurines under mild coupling conditions [cat. 4-dimethylaminopyridine (DMAP) and excess methyl trimethylsilyl dimethylketene acetal (MTDA) as a proton trap].

Full text of DOI:10.1016/0040-4039(96)01963-6

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Product name:((S)-1-Chlorosulfonylmethyl-2-phenyl-ethyl)-carbamic acid tert-butyl ester

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