Synthesis of 3-fluoro azetidinone by electrophilic fluorination

DOI: 10.1016/S0040-4039(96)02217-4

Source and publish data:

Tetrahedron Letters p. 69 - 72 (1997)

Update date:2022-09-26

Topics:

Authors:

Genet, Jean-Pierre

Durand, Jean-Olivier

Roland, Sylvain

Savignac, Monique

Jung, Frederic

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Article abstract of DOI:10.1016/S0040-4039(96)02217-4

An easy access to the 3-fluoroazetidinone 4a based on electrophilic fluorination, is reported. The fluorination of the β-lactam 7 with Differding's N-fluorosulfonimide proceeds stereoselectively, under mild conditions and in good yield.

Full text of DOI:10.1016/S0040-4039(96)02217-4

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