Synthesis of enantiopure (nor)-azatropanes via N-acylhydrazonium ion intermediates

DOI: 10.1016/S0040-4039(96)02241-1

Source and publish data:

Tetrahedron Letters p. 155 - 158 (1997)

Update date:2022-08-05

Topics:

Authors:

Teerhuis, N. Miranda

Hiemstra, Henk

Speckamp, W. Nico

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Article abstract of DOI:10.1016/S0040-4039(96)02241-1

The synthesis of a number of aza-analogues of (nor)tropanes is described. Key features of the synthesis include the efficient preparation of an enantiopure 5-substituted 3-pyrazolidinone and stereoselective cyclization of an N-acylhydrazonium ion intermediate.

Full text of DOI:10.1016/S0040-4039(96)02241-1

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