Ring expansions of tetrahydroprotoberberines and related dibenzo[c,g]azecines modulate the dopamine receptor subtype affinity and selectivity

DOI: 10.1002/ardp.200900267

Source and publish data:

Archiv der Pharmazie p. 207 - 214 (2010)

Update date:2022-07-29

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Authors:

Schulze, Maria

Siol, Oliver

Meise, Werner

Lehmann, Jochen

Enzensperger, Christoph

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Article abstract of DOI:10.1002/ardp.200900267

The affinities of tetrahydroprotoberberines for dopamine receptors dramatically decrease after cleaving the central C-N bond to the analogous ten-membered dibenzo[c,g]azecines [1]. In the present work, we also synthesized eleven-membered homologues of the

Full text of DOI:10.1002/ardp.200900267

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