Fluorinated peptides incorporating a 4-fluoroproline residue as potential inhibitors of HIV protease

DOI: 10.1016/S0022-1139(96)03568-3

Source and publish data:

Journal of Fluorine Chemistry p. 125 - 130 (1997)

Update date:2022-08-03

Topics:

Authors:

Tran, Thanh Thu

Patino, Nadia

Condom, Roger

Frogier, Tea

Guedj, Roger

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Article abstract of DOI:10.1016/S0022-1139(96)03568-3

N-Fmoc-4-fluoro-L-proline methyl ester was prepared as an attractive synthon for both solid and solution phase peptide synthesis. Its use for the synthesis of Fmoc-Phe-Pro(F)-OMe and Fmoc-Pro(F)-Val-Val-OMe is presented. Direct fluorination with DAST of a

Full text of DOI:10.1016/S0022-1139(96)03568-3

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