Incorporation of conformationally constrained phenylalanine derivatives TIC, SIC, HIC and NIC into a cholecystokinin-B/gastrin receptor antagonist

DOI: 10.1016/S0960-894X(97)00211-4

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 1289 - 1292 (1997)

Update date:2022-08-04

Topics:

Authors:

Gibson, Susan E.

Guillo, Nathalie

Kalindjian, S. Barret

Tozer, Matthew J.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0960-894X(97)00211-4

The preparation and biological properties of a conformationally constrained series of cholecystokinin-B/gastrin receptor ligands are described. The membered ring (Nic) derivative was found to be as active at these receptors as an unconstrained phenylalani

Full text of DOI:10.1016/S0960-894X(97)00211-4

Products guided by the article

Product name:1,3-Benzenedicarboxylic acid, 5-[[(1,2,3,4-tetrahydro-3-isoquinolinyl)carbonyl]amino]-, bis(phenylmethyl) ester

Cas No:192133-89-4

R&D Labs maybe for 192133-89-4

Guangzhou Puho Pharmaceutical Technology Co. Ltd.

Contact:86-20-29848035/29848075

Address:No.166, Chaoyang East Road, Panyu District, Guangzhou City, Guangdong Province
X.T.Y Environ-Tech Co.,Ltd

Contact:+86-310-7092106

Address:Quzhou Modern & New Industrial Park, Handan, Hebei 057250, China
KODI CHEMICAL CO., LTD

Contact:021

Address:Pudong
KA-SHING Business Trade Macau Co., Ltd.

Contact:00853-28430045

Address:23rd Floor, Block 3 La Cite, Areia Preta, Macao
Weifang Ocean Trading Co., Ltd.

Contact:+86-536-2081155

Address:Room2606, Yuqing Building, 518#, Yuquan Road, High-tech Development Zone, Weifang City, Shandong Province, China

Relevant to this article

Synthesis of a versatile multifunctional building block for the construction of polyketide natural products containing ethyl side-chains

Doi:10.1039/b610702h
(2006)
Novel synthetic approaches to monocyclic β-lactam antibiotics

Doi:10.1002/bscb.19840930705
(1984)
4′-Alkoxyl substitution enhancing the anti-mitotic effect of 5-(3′,4′,5′-substituted)anilino-4-hydroxy-8-nitroquinazolines as a novel class of anti-microtubule agents

Doi:10.1016/j.bmcl.2006.08.058
(2006)
'O-Acyl isopeptide method': racemization-free segment condensation in solid phase peptide synthesis

Doi:10.1016/j.tetlet.2006.09.001
(2006)
Doi:10.1021/ja01154a102
(1951)
A practical one-pot procedure for the synthesis of pyrazino[2′,3′:4,5]thieno[3,2-d]pyrimidinones by a tandem aza-Wittig/heterocumulene-mediated annulation strategy

Doi:10.1016/j.tet.2006.09.028
(2006)

Article Doi