Incorporation of conformationally constrained phenylalanine derivatives TIC, SIC, HIC and NIC into a cholecystokinin-B/gastrin receptor antagonist

DOI: 10.1016/S0960-894X(97)00211-4

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 1289 - 1292 (1997)

Update date:2022-08-04

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Authors:

Gibson, Susan E.

Guillo, Nathalie

Kalindjian, S. Barret

Tozer, Matthew J.

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Article abstract of DOI:10.1016/S0960-894X(97)00211-4

The preparation and biological properties of a conformationally constrained series of cholecystokinin-B/gastrin receptor ligands are described. The membered ring (Nic) derivative was found to be as active at these receptors as an unconstrained phenylalani

Full text of DOI:10.1016/S0960-894X(97)00211-4

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Product name:1,3-Benzenedicarboxylic acid, 5-[[(1,2,3,4-tetrahydro-3-isoquinolinyl)carbonyl]amino]-, bis(phenylmethyl) ester

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