A synthetic route for the generation of C-7 substituted azepinones

DOI: 10.1016/S0040-4039(00)76227-7

Source and publish data:

Tetrahedron Letters p. 1393 - 1396 (1994)

Update date:2022-08-03

Topics:

Authors:

Robl, Jeffrey A.

Cimarusti, Maria P.

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Article abstract of DOI:10.1016/S0040-4039(00)76227-7

A versatile method for the synthesis of 3-amino azepinones possessing alkyl substitution at the C-7 position is described. Compounds of this type may be viewed as conformationally restricted dipeptide surrogates.

Full text of DOI:10.1016/S0040-4039(00)76227-7

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