
Bioorganic and Medicinal Chemistry Letters p. 2409 - 2414 (1997)
Update date:2022-08-03
Topics:
Li, Pui-Kai
Chu, Guo-Hua
Gillen, Megan L.
Parekh, Tejal
Witt-Enderby, Paula A.
We report the synthesis and radioligand binding analysis of a novel charged melatonin receptor ligand, N-[2-(2-Trimethylammoniumethyleneoxy-7-methoxy)ethyl] propionamide iodide. The charged ligand has potential in determining whether internalization of th
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