Asymmetric synthesis of L-azetidine-2-carboxylic acid and 3-substituted congeners - Conformationally constrained analogs of phenylalanine, naphthylalanine, and leucine

DOI: 10.1016/S0960-894X(99)00218-8

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 1437 - 1442 (1999)

Update date:2022-08-04

Topics:

Authors:

Hanessian, Stephen

Bernstein, Naomy

Yang, Rui-Yang

Maguire, Robert

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0960-894X(99)00218-8

Enantiopure L-azetidine-2-carboxylic acid, the (3R)-phenyl, (3R)- naphthyl and (3S)-isopropyl analogs were prepared based on a zinc-mediated asymmetric addition of allylic halides to the camphor sultam derivative of glyoxylic acid O-benzyl oxime.

Full text of DOI:10.1016/S0960-894X(99)00218-8

Products guided by the article

Product name:(2S,3S)-2-Benzyloxyamino-1-((1S,5R,7R)-10,10-dimethyl-3,3-dioxo-3λ⁶-thia-4-aza-tricyclo[5.2.1.0^1,5]dec-4-yl)-3-naphthalen-1-yl-pent-4-en-1-one

Cas No:231609-73-7

R&D Labs maybe for 231609-73-7

Jinan Decheng Hemu Medical Technology Co.，Ltd.

Contact:+86-531-68650525

Address:NO.554 Zhengfeng Road High-new Technology Development Zone
Taixing Joxin Bio-tec Co.,Ltd.

website:http://www.joxbio.com

Contact:86-523-87558858 87612088

Address:No.88, chengdong industrial park
Puyang Huicheng Electronic Material Co., Ltd

website:http://huichengchem.weba.testwebsite.cn/index_en.html

Contact:+86-393-8910800

Address:West Section Shengli Road, Puyang457000, China
TLS PHARMACEUTICAL CO.,LTD

Contact:0833-5590788/5590338/5590055

Address:Victory in the town of Red Star Village,Mount Emei City,industrial concentration area storage processing logistics parkpark
Jiangsu Haian Petro chemical Plant

Contact:+86-513-88902723

Address:99, Changjiang West Road, Haian County, Jiangsu

Relevant to this article

One-pot synthesis of 2,3-disubstituted naphtho[2,3-b]thiophene-4,9-diones from a 2-sulfenyl-1,4-naphthoquinone and enamines

Doi:10.1246/cl.1999.503
(1999)
Chemical Control of Mammalian Circadian Behavior through Dual Inhibition of Casein Kinase Iα and δ

Doi:10.1021/acs.jmedchem.8b01541
(2019)
Synthesis and equilibrium studies of mixed-ligand complexes of Co(II), Ni(II), and Cu(II) with some aliphatic dicarboxylic acids and creatinine

Doi:10.1081/SIM-120030438
(2004)
Studies on chemical carcinogens. 8. The structure-carcinogenicity relationship among derivatives of 4-nitro- and 4-hydroxyamino-quinoline 1-oxides (supplement).

Doi:10.1248/cpb.17.544
(1969)
Synthesis of acetyl scopine. Intramolecular reactions of N-carbethoxy nortropine-3α-benzene-sulfenate

Doi:10.1055/s-1999-2658
(1999)
Effects of mixed H₂O-CH₃CN solvents on the Bronsted coefficient for the intramolecular general base-catalyzed cleavage of ionized phenyl salicylate in the presence of primary and secondary amines

Doi:10.1002/(SICI)1097-4601(2000)32:3<153::AID-KIN5>3.0.CO;2-W
(2000)

Article Doi