Bioorganic and Medicinal Chemistry Letters p. 2955 - 2958 (2001)
Update date:2022-08-04
Topics:
Wattanasin, Sompong
Weidmann, Beat
Roche, Didier
Myers, Stewart
Xing, Amy
Guo, Qin
Sabio, Michael
Von Matt, Peter
Hugo, Ronald
Maida, Susan
Lake, Philip
Weetall, Marla
The synthesis and identification of a novel series of inhibitors of integrin VLA-4 are described. Their in vitro activity and selectivity against closely related integrins are also presented.
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Doi:10.1039/a902196e
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