European Journal of Medicinal Chemistry p. 495 - 507 (2018)
Update date:2022-09-26
Topics:
Ahonen, Tiina J.
Rinne, Maiju
Grutschreiber, Peter
M?tlik, Kert
Airavaara, Mikko
Schaarschmidt, Dieter
Lang, Heinrich
Reiss, David
Xhaard, Henri
Gaveriaux-Ruff, Claire
Yli-Kauhaluoma, Jari
Moreira, Vania M.
Despite extensive years of research, the direct oxidation of the 7,8-double bond of opioids has so far received little attention and knowledge about the effects of this modification on activity at the different opioid receptors is scarce. We herein report
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