Synthesis of the peptidic α-hydroxy amides phebestin, probestin, and bestatin from α-keto amide precursors

DOI: 10.1016/S0040-4039(99)01143-0

Source and publish data:

Tetrahedron Letters p. 6163 - 6166 (1999)

Update date:2022-07-31

Topics:

Authors:

Wasserman, Harry H.

Xia, Mingde

Petersen, Anders K.

Jorgensen, Michael R.

Curtis, Erin A.

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Article abstract of DOI:10.1016/S0040-4039(99)01143-0

Aminopeptidase inhibitors, phebestin, probestin and bestatin have been prepared by stereospecific reduction of α-keto amide precursors using zinc borohydride.

Full text of DOI:10.1016/S0040-4039(99)01143-0

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