Novel 1,4-naphthoquinone-based sulfonamides: Synthesis, QSAR, anticancer and antimalarial studies

DOI: 10.1016/j.ejmech.2015.09.001

Source and publish data:

European Journal of Medicinal Chemistry p. 446 - 459 (2015)

Update date:2022-08-15

Topics: Synthesis QSAR (quantitative structure-activity relationship)

Authors:

Pingaew, Ratchanok

Prachayasittikul, Veda

Worachartcheewan, Apilak

Nantasenamat, Chanin

Prachayasittikul, Supaluk

Ruchirawat, Somsak

Prachayasittikul, Virapong

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Article abstract of DOI:10.1016/j.ejmech.2015.09.001

A novel series of 1,4-naphthoquinones (33-44) tethered by open and closed chain sulfonamide moieties were designed, synthesized and evaluated for their cytotoxic and antimalarial activities. All quinone-sulfonamide derivatives displayed a broad spectrum o

Full text of DOI:10.1016/j.ejmech.2015.09.001

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