Aminotetralins as narcotic antagonists. 2. Synthesis and opiate-related activity of 1-phenyl-3-aminotetralins

DOI: 10.1021/jm00345a005

Source and publish data:

Journal of Medicinal Chemistry p. 216 - 220 (1982)

Update date:2022-08-04

Topics: Synthesis Narcotic Antagonists

Authors:

Fries Fries

Bertelli

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00345a005

The synthesis and analgetic agonist and antagonist activities of several 3-[N-(cyclopropylmethyl)-N-methylamino]-1-phenyltetralins are reported. The design of these agents was based partially on the possibility of two aryl receptor binding sites on the op

Full text of DOI:10.1021/jm00345a005

Products guided by the article

Product name:ethyl 3-(methylamino)-4-phenylbutyrate

Cas No:60546-98-7

R&D Labs maybe for 60546-98-7

Jiangxi Hito Chemical Co., Ltd.

Contact:+86-792-3170318

Address:No. 6, Tianhong Ave., Xinghuo Industry Park, Yongxiu, Jiujiang, Jiangxi, China
Beijing Harmony Chemical Co., Ltd.

Contact:86-010-84956928

Address:Room 207, Jin feng he B building, No 8 Xin Jie Kou Wai Street, Xi Cheng District, Beijing,PRC. 10008
Wuxi Pharma-Trading Import & Export Co.,Ltd.

Contact:+86-510-82304590 82716390

Address:Room 523,Youzu Alliance Building,No.88 Renmin Zhonglu,Wuxi,Jiangsu,China
Shanghai Apeptide Co., Ltd.

website:http://www.apeptides.com/en/

Contact:+86-21-60871011

Address:No. 80 Chuanshan Shuyuan Steet,Pudong,Shanghai
Anqing World Chemical Co., Ltd.

Contact:+86-556-5800026

Address:Daguan Economic Development Zone of circular economy industrial park Anqing City Anhui province

Relevant to this article

4-Aminophenyldiphenylphosphinite (APDPP), a new heterogeneous and acid scavenger phosphinite - Conversion of alcohols, trimethylsilyl, and tetrahydropyranyl ethers to alkyl halides with halogens or N-halosuccinimides

Doi:10.1139/V06-120
(2006)
Synthesis and biological evaluation of menthol-based derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1)

Doi:10.1016/S0960-894X(03)00686-3
(2003)
Nylon/DNA: Single-stranded DNA with a covalently stitched nylon lining

Doi:10.1021/ja035186r
(2003)
Doi:10.1021/jo00817a036
(1971)
The identification of a novel highly condensed pentacyclic heteroaromatic ring system 1,3,5,5b,6,8,10,10b-octaazacyclopenta[h,i]aceanthrylene and its application in the synthesis of 5,7-substituted pyrazolo[4,3-d]pyrimidines

Doi:10.1002/jhet.2147
(2015)
Doi:10.1021/ja00433a048
(1976)

Article Doi