Regioselective iodoamination of terminal ynamides for the synthesis of α-amino-β,β-diiodo-enamides

Article abstract of DOI:10.1039/c6cc00370b

A mild and efficient methodology involving the I₂/TBHP-mediated intermolecular iodoamination of ynamides with amines for the synthesis of α-amino-β,β-diiodo-enamides was developed. This reaction provides the first intermolecular iodoamination o