Synthesis, conformation, and dopaminergic activity of 5,6-ethano-bridged derivatives of selective dopaminergic 3-benzazepines

Article abstract of DOI:10.1021/jm00391a007

To probe the suggestion that D-1 (DA₁) dopamine receptors might possess an accessory π-binding site in a location complementary to a suitably oriented aromatic ring (i.e., in an axial orientation approximately orthogonal to the catechol nucleus