Bioorganic and Medicinal Chemistry Letters p. 1486 - 1490 (2006)
Update date:2022-09-26
Topics:
Alper, Phillip B.
Liu, Hong
Chatterjee, Arnab K.
Nguyen, Khanhlinh T.
Tully, David C.
Tumanut, Christine
Li, Jun
Harris, Jennifer L.
Tuntland, Tove
Chang, Jonathan
Gordon, Perry
Hollenbeck, Thomas
Karanewsky, Donald S.
A systematic study of anilines led to the discovery of a metabolically robust fluoroindoline replacement for the alkoxy aniline toxicophore in 1. Investigations of the P1 pocket resulted in the discovery of a wide tolerance of functionality leading to the discovery of 11 as a potent and selective inhibitor of cathepsin S.
View MoreLIAOYANG WANRONG CHEMICALS COMPANY LIMITED
Contact:86-419-2390789
Address:XINLI VILLAGE , DONG NINGWEI COUNTY,TAIZIHE DISTRICT, LIAOYANG , LIAONING
Hangzhou Gangjin Chemical Co.,Ltd.(expird)
Contact:+86-571-85109780
Address:707 Zhejiang Minhang Bldg., No.290 Zhongshan North Road, Hangzhou 310003, China
Contact:86-311-83160559
Address:shijiazhuang
jintan yufan Medicine Raw materials Co.,Ltd.(expird)
Contact:86-519-82808282
Address:6th,Jincheng Huangzhuang
Disynthesis Chemical Technology Co. Ltd.
Contact:+86-571-88194596
Address:Dengyun road 380, Gongshu district, Hangzhou city, China
Doi:10.1016/S0040-4039(00)78707-7
(1980)Doi:10.1080/00397910902788125
(2009)Doi:10.1021/jm950117b
(1996)Doi:10.1016/S0040-4039(00)78687-4
(1980)Doi:10.1021/acscatal.8b01897
(2018)Doi:10.1039/c4ob00938j
(2014)