Journal of Medicinal Chemistry p. 559 - 567 (1981)
Update date:2022-08-04
Topics:
Rosowsky, Andre
Yu, Cheng-Sein
Uren, Jack
Lazarus, Herbert
Wick, Michael
Carbodiimide-mediated condensation of 4-amino-4-deoxy-N10-methylpteroic acid (APA) with several alkyl, aralkyl, and aryl amines, in the presence or absence of N-hydroxysuccinimide, was employed in order to prepare new lipid-soluble bis(amide) d
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