Bioorganic and Medicinal Chemistry Letters p. 814 - 818 (2007)
Update date:2022-07-30
Topics:
Meyers, Kenneth M.
Kim, Nicholas
Mendez-Andino, Jose L.
Hu, X. Eric
Mumin, Rashid N.
Klopfenstein, Sean R.
Wos, John A.
Mitchell, Maria C.
Paris, Jennifer L.
Ackley, David C.
Holbert, Jerry K.
Mittelstadt, Scott W.
Reizes, Ofer
Aminomethyl tetrahydronaphthalene biphenyl carboxamide MCH-R1 antagonists with greater selectivity over hERG were identified. SAR studies addressing two distinct alternatives for structural modifications leading to improve hERG selectivity are described.
View MoreJinan Hongfangde Pharmatech Co.LTD
Contact:0531-88870908
Address:F Bldg,750#,Shunhua Rd,New&High-tech Zone,Jinan,Shandong,China 250101
Jiangxi Huashi Pharmaceutical Co., Ltd
Contact:+86-795-4509628
Address:Ningbo Ave., Fengtian Industrial Park, Fengxin Country, Jiangxi, China.
Chengdu Sino-Strong Pharmaceutical Co.,Ltd.
website:http://www.sino-strong.com.cn
Contact:+86-28-82666753
Address:459 West haike road,Cross-straits technological industry park, Wenjiang district,Chengdu, P.R.China
Refine Chemicals Science & Technology Technology Developing Co., Ltd.
Contact:+86-22-87899130
Address:No.12,west keyan road,Tianjin City
Shenzhen HwaGen Pharmaceutical Co., Ltd
website:http://www.rafflespt.com
Contact:+86-752-5538396
Address:Guangdong Huizhou China
Doi:10.1021/jo0478196
(2005)Doi:10.1021/om0490583
(2005)Doi:10.1016/S0020-1693(00)90258-5
(1982)Doi:10.1039/P19840000583
(1984)Doi:10.1021/ja047437h
(2005)Doi:10.1021/jm1008659
(2011)