Bioorganic and Medicinal Chemistry Letters p. 814 - 818 (2007)
Update date:2022-07-30
Topics:
Meyers, Kenneth M.
Kim, Nicholas
Mendez-Andino, Jose L.
Hu, X. Eric
Mumin, Rashid N.
Klopfenstein, Sean R.
Wos, John A.
Mitchell, Maria C.
Paris, Jennifer L.
Ackley, David C.
Holbert, Jerry K.
Mittelstadt, Scott W.
Reizes, Ofer
Aminomethyl tetrahydronaphthalene biphenyl carboxamide MCH-R1 antagonists with greater selectivity over hERG were identified. SAR studies addressing two distinct alternatives for structural modifications leading to improve hERG selectivity are described.
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