Journal of Medicinal Chemistry p. 10848 - 10866 (2019)
Update date:2022-08-15
Topics: in vivo Agonists Histamine H3 receptor Non-imidazole 4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines High-Affinity Central Nervous System Activity
Wágner, Gábor
Mocking, Tamara A. M.
Arimont, Marta
Provensi, Gustavo
Rani, Barbara
Silva-Marques, Bruna
Latacz, Gniewomir
Da Costa Pereira, Daniel
Karatzidou, Christina
Vischer, Henry F.
Wijtmans, Maikel
Kie?-Kononowicz, Katarzyna
De Esch, Iwan J. P.
Leurs, Rob
Despite the high diversity of histamine H3 receptor (H3R) antagonist/inverse agonist structures, partial or full H3R agonists have typically been imidazole derivatives. An in-house screening campaign intriguingly afforded
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