Structure-activity relationships of C-terminal tri- and tetrapeptide fragments that inhibit gastrin activity

Article abstract of DOI:10.1021/jm00381a002

A series of tri- and tetrapeptide derivatives, analogues of the gastrin C-terminal region with no phenylalanine residue, were synthesized. These peptides were tested for their ability to inhibit gastrin-stimulated acid secretion in vivo as well as binding