Synthesis and Some Pharmacological Properties of 18 Potent O-Alkyltyrosine-Substituted Antagonists of the Vasopressor Responses to Arginine-Vasopressin

DOI: 10.1021/jm00148a019

Source and publish data:

Journal of Medicinal Chemistry p. 1485 - 1491 (1985)

Update date:2022-08-03

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Authors:

Manning, Maurice

Lammek, Bernard

Bankowski, Krzysztof

Seto, Janny

Sawyer, W. H.

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Article abstract of DOI:10.1021/jm00148a019

Using the Merrifield solid-phase method, we have synthesized 18 new 2-O-alkyltyrosine-substituted analogues (where alkyl = methyl and ethyl) of the arginine-vasopressin (AVP) vasopressor antagonists <1-deaminopenicillamine>arginine-vasopressin (dPAVP), <1

Full text of DOI:10.1021/jm00148a019

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Product name:<1-deaminopenicillamine,2-O-ethyltyrosine,4-valine>arginine-vasopressin

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