TIPP: A Highly Potent and Stable Pseudopeptide δ Opioid Receptor Antagonist with Extraordinary δ Selectivity

DOI: 10.1021/jm00073a020

Source and publish data:

Journal of Medicinal Chemistry p. 3182 - 3187 (1993)

Update date:2022-08-11

Topics:

Authors:

Schiller, Peter W.

Weltrowska, Grazyna

Nguyen, Thi M.-D.

Wilkes, Brian C.

Chung, Nga N.

Lemieux, Carole

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Article abstract of DOI:10.1021/jm00073a020

Pseudopeptide analogues of the δ opioid antagonists H-Tyr-Tic-Phe-Phe-OH (TIPP) and H-Tyr-Tic-Phe-OH (TIP) containing a reduced peptide bond between the Tic² and Phe³ residues were synthesized.The two compounds, H-Tyr-TicψPhe-

Full text of DOI:10.1021/jm00073a020

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