Journal of Medicinal Chemistry p. 4087 - 4102 (2018)
Update date:2022-08-15
Topics:
García-Reyes, Balbina
Witt, Lydia
Jansen, Bj?rn
Karasu, Ebru
Gehring, Tanja
Leban, Johann
Henne-Bruns, Doris
Pichlo, Christian
Brunstein, Elena
Baumann, Ulrich
Wesseler, Fabian
Rathmer, Bernd
Schade, Dennis
Peifer, Christian
Knippschild, Uwe
Inhibitors of Wnt production (IWPs) are known antagonists of the Wnt pathway, targeting the membrane-bound O-acyltransferase porcupine (Porcn) and thus preventing a crucial Wnt ligand palmitoylation. Since IWPs show structural similarities to benzimidazol
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