Bioorganic and Medicinal Chemistry Letters p. 1381 - 1384 (2000)
Update date:2022-08-11
Topics:
Collins, Ian
Davey, William B.
Rowley, Michael
Quirk, Kathleen
Bromidge, Frances A.
McKernan, Ruth M.
Thompson, Sally-Anne
Wafford, Keith A.
A new class of N-(indol-3-ylglyoxylyl)piperidines are high affinity agonists at the benzodiazepine binding site of human GABA-A receptor ion-channels, with modest selectivity for receptors containing the α1 subunit over α2 and α3. All three receptor subtypes discriminate substantially between the two enantiomers of the chiral ligand 10. (C) 2000 Elsevier Science Ltd. All rights reserved.
View MoreShanghai He Yang International Trading Co., Ltd.
Contact:+86-21-52043598
Address:Room 816, Blag.5, No.58 Huachi Road
Contact:+86-18653358619
Address:zibo
Wuhan Chemchemical Co., Ltd.(expird)
Contact:15973022782
Address:7-5-6218,Incubation Centre,Guandong Industry Park, East Lake High-Tech Development Zone,Wuhan City.
Fuxin Jintelai Fluorin Chemical Co., Ltd.
Contact:+86-0418-8229599
Address:, 7th Huagong Road, Fluorine industry development zone (Yimatu Town,Fumeng County),Fuxin City, Liaoning Province, China
Jining tiansheng chemical co.,ltd.
Contact:+86-537-5158722
Address:ROOM 1011, BLOCK B, CUIDU INTERNATIOAL BUSINESS CENTER, JINING CITY, CHINA
Doi:10.1021/jo9622338
(1997)Doi:10.1039/c5gc02494c
(2016)Doi:10.1080/00397910802219569
(2008)Doi:10.2478/s11696-011-0066-6
(2011)Doi:10.1016/0031-9422(96)00191-4
(1996)Doi:10.1016/S0040-4039(02)00376-3
(2002)
