Conformationally constrained nonpeptide β-turn mimetics of enkephalin

DOI: 10.1016/S0040-4020(01)90205-4

Source and publish data:

Tetrahedron p. 3433 - 3448 (1993)

Update date:2022-08-03

Topics:

Authors:

Gardner, Benjamin

Nakanishi, Hiroshi

Kahn, Michael

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Article abstract of DOI:10.1016/S0040-4020(01)90205-4

The design, synthesis and in vitro biological analysis of a family of conformationally constrained nonpeptide mimetics incorporating a 4→1 β-turn prosthetic unit to examine the proposed biological significance of this conformer is described.

Full text of DOI:10.1016/S0040-4020(01)90205-4

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