
Angewandte Chemie - International Edition p. 9279 - 9283 (2021)
Update date:2022-08-04
Topics: Selective Development Experimental Plasmodium falciparum
Zhan, Wenhu
Zhang, Hao
Ginn, John
Leung, Annie
Liu, Yi J.
Michino, Mayako
Toita, Akinori
Okamoto, Rei
Wong, Tzu-Tshin
Imaeda, Toshihiro
Hara, Ryoma
Yukawa, Takafumi
Chelebieva, Sevil
Tumwebaze, Patrick K.
Lafuente-Monasterio, Maria Jose
Martinez-Martinez, Maria Santos
Vendome, Jeremie
Beuming, Thijs
Sato, Kenjiro
Aso, Kazuyoshi
Rosenthal, Philip J.
Cooper, Roland A.
Meinke, Peter T.
Nathan, Carl F.
Kirkman, Laura A.
Lin, Gang
Plasmodium falciparum proteasome (Pf20S) inhibitors are active against Plasmodium at multiple stages—erythrocytic, gametocyte, liver, and gamete activation stages—indicating that selective Pf20S inhibitors possess the potential to be therapeutic, prophyla
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