SYNTHESIS OF THE DIASTEREOMERIC 2-ARYL-1-CYCLOHEXYL-3-(2,3-EPOXYPROPIONYL)AZIRIDINES

Article abstract of DOI:10.1007/BF00542772

The reaction of cinnamoyloxiranes with an iodine cyclohexylamine complex in the presence of an excess of amine led to a mixture of the four diastereomeric epoxypropionylaziridines the ratio of which depended on steric and electronic factors in the substrate and reactants.