
European Journal of Medicinal Chemistry p. 91 - 100 (1987)
Update date:2022-08-05
Topics:
Blakemore, Robert C.
Ganellin, C. Robin
Garbarg, Monique
Gros, Claude
Ife, Robert J.
et al.
The synthesis is described of potential I-labelled H1-receptor ligands.Receptor affinity is assessed in vitro from inhibition of histamine-stimulated contraction of guinea pig ileum and/or through binding to guinea pig cerebellar membranes.Dire
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