Bioorganic and Medicinal Chemistry Letters p. 3669 - 3673 (2009)
Update date:2022-08-02
Topics:
Charrier, Nicolas
Clarke, Brian
Demont, Emmanuel
Dingwall, Colin
Dunsdon, Rachel
Hawkins, Julie
Hubbard, Julia
Hussain, Ishrut
Maile, Graham
Matico, Rosalie
Mosley, Julie
Naylor, Alan
O'Brien, Alistair
Redshaw, Sally
Rowland, Paul
Soleil, Virginie
Smith, Kathrine J.
Sweitzer, Sharon
Theobald, Pam
Vesey, David
Walter, Daryl S.
Wayne, Gareth
Our first generation of hydroxyethylamine transition-state mimetic BACE-1 inhibitors allowed us to validate BACE-1 as a key target for Alzheimer's disease by demonstrating amyloid lowering in an animal model, albeit at rather high doses. Finding a molecul
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