
Organic Letters p. 1027 - 1029 (2009)
Update date:2022-08-03
Topics:
Xu, Xiaoliang
Li, Xiaonian
Mediated by copper/diethyl azodicarboxylate, regioselective alkynylation of unactivated aliphatic tertiary methylamine with terminal alkyne was successfully established. It is not necessary for the tertiary methylamines to be aryl substituted to modulate
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