Synthesis and Structure-Activity Relationships of a Novel Series of Non-Peptide Angiotensin II Receptor Binding Inhibitors Specific for the AT2 Subtype

DOI: 10.1021/jm00115a014

Source and publish data:

Journal of Medicinal Chemistry p. 3248 - 3260 (1991)

Update date:2022-07-29

Topics:

Authors:

Blankley, C. John

Hodges, John C.

Klutchko, Sylvester R.

Himmelsbach, Richard J.

Chucholowski, Alexander

et al. et al.

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Article abstract of DOI:10.1021/jm00115a014

Structure-activity relationships are reported for a novel class of 4,5,6,7-tetrahydro-1H-imidazo<4,5-c>pyridine-6-carboxylic acid derivatives that displace 125I-labeled angiotensin II from a specific subset of angiotensin II (Ang II) binding sites in rat

Full text of DOI:10.1021/jm00115a014

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