Synthesis of 1,5-diaryl-3-methyl-1H-pyrazolo[4,5-c]isoquinolines and studies of binding to specific peripheral benzodiazepine binding sites

DOI: 10.1002/jps.2600780602

Source and publish data:

Journal of Pharmaceutical Sciences p. 437 - 442 (1989)

Update date:2022-07-29

Topics:

Authors:

Cecchi Cecchi

Colotta Colotta

Melani Melani

Palazzino

Filacchioni

Martini Martini

Giannaccini

Lucacchini

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Article abstract of DOI:10.1002/jps.2600780602

Some 1,5-diaryl-3-methyl-1H-pyrazolo[4,5-c]isoquinolines were synthesized and tested for their ability to displace [³H]clonazepam or [³H]Ro 5-4864 from their specific binding on the central and peripheral benzodiazepine receptors. No

Full text of DOI:10.1002/jps.2600780602

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